SCHEMBL11005537

SCHEMBL11005537

C#CCNc1ccc(-c2nc3cncnc3[nH]2)c(OC)c1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 15/20 0.39
PDE5A O76074 2/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
PDE7A Q13946 1/20 0.35
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11011479 0.92 AMY1A (0.34) CYP17A1PDE5A
SCHEMBL11010174 0.89 CYP17A1 (0.39) CYP17A1PDE5APDE3BPDE3APDE7A
SCHEMBL11005543 0.84 ENPP1 (0.46) CYP17A1PDE5APDE3BPDE3A
SCHEMBL11009498 0.84 PDE10A (0.38) CYP17A1PDE5APDE3BPDE3APDE7A
SCHEMBL11008331 0.83 ENPP1 (0.41) CYP17A1PDE5APDE3BPDE3APDE7A
SCHEMBL11004488 0.83 MAOB (0.40) PDE5APDE3BPDE3A
SCHEMBL11010059 0.82 CYP17A1 (0.40) CYP17A1PDE5APDE3BPDE3A
SCHEMBL11010093 0.81 PDE5A (0.35) CYP17A1PDE5APDE3BPDE3AAAK1
SCHEMBL11009966 0.81 PIK3CD (0.35) CYP17A1PDE5A
SCHEMBL11009531 0.81 PDE5A (0.35) CYP17A1PDE5APDE3BPDE3AAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed