SCHEMBL11009397

SCHEMBL11009397

C=CCSc1ccc(-c2nc3cncnc3[nH]2)c(OC)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
AMY1A P0DUB6 6/20 0.33
ENPP1 P22413 1/20 0.33
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PDE2A O00408 1/20 0.32
CHEK2 O96017 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
CYP17A1 P05093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11010240 0.93 AMY1A (0.34) PDE5AAMY1AENPP1NPC1ALDH1A1
SCHEMBL11009297 0.84 PDE5A (0.35) PDE5APDE3BPDE3AAMY1AENPP1
SCHEMBL11003382 0.84 EGFR (0.31)
SCHEMBL11010093 0.84 PDE5A (0.35) PDE5APDE3BPDE3AAMY1AENPP1
SCHEMBL11009401 0.84 ENPP1 (0.43) PDE5APDE3BPDE3AAMY1AENPP1
SCHEMBL11012150 0.83 HPGD (0.42) PDE5APDE3BPDE3AENPP1ALDH1A1
SCHEMBL9634366 0.82 PDE5A (0.47) PDE5APDE3BPDE3AAMY1AENPP1
SCHEMBL11012358 0.81 SMN1; SMN2 (0.41) PDE5APDE3BPDE3ANPC1ALDH1A1
SCHEMBL11009498 0.80 PDE10A (0.38) PDE5APDE3BPDE3ANPC1ALDH1A1
SCHEMBL10740548 0.80 PDE2A (0.42) PDE5APDE3BPDE3AENPP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed