SCHEMBL1101

SCHEMBL1101

Cc1c(CN2CCc3c(c4ccccc4n3C)C2=O)ncn1S(=O)(=O)N(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.60
HTR2B P41595 4/20 0.60
CYP3A4 P08684 3/20 0.60
HTR2A P28223 3/20 0.60
HTR2C P28335 3/20 0.60
CYP1A2 P05177 2/20 0.60
HTR3A P46098 2/20 0.60
ADRA2C P18825 1/20 0.60
ADRA1A P35348 1/20 0.60
CASP6 P55212 1/20 0.59
CYP2D6 P10635 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
SLC22A2 O15244 1/20 0.36
SLC22A1 O15245 1/20 0.36
SLC22A3 O75751 1/20 0.36
HTR3B O95264 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7286786 0.86 KCNH2 (0.44) KCNH2HTR2BCYP3A4HTR2AHTR2C
SCHEMBL9485681 0.86 KCNH2 (0.44) KCNH2HTR2BCYP3A4HTR2AHTR2C
SCHEMBL10123935 0.82 KCNH2 (0.66) KCNH2HTR2BCYP3A4HTR2AHTR2C
SCHEMBL7375451 0.81 KCNH2 (0.55) KCNH2HTR2BCYP3A4HTR2AHTR2C
SCHEMBL10108911 0.81 KCNH2 (0.64) KCNH2HTR2BCYP3A4HTR2AHTR2C
SCHEMBL1484 0.79 KCNH2 (0.62) KCNH2HTR2BCYP3A4HTR2AHTR2C
SCHEMBL9597563 0.79 KCNH2 (0.52) KCNH2HTR2BCYP3A4HTR2AHTR2C
Fumaric Acid SCHEMBL9676 0.78 KCNH2 (0.60) KCNH2HTR2BCYP3A4HTR2AHTR2C
Maleic Acid SCHEMBL9675 0.78 KCNH2 (0.60) KCNH2HTR2BCYP3A4HTR2AHTR2C
Alosetron SCHEMBL850 0.76 KCNH2 (0.90) KCNH2HTR2BCYP3A4HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360800-A Tetrahydro-1H-pyrido[4,3-b]indol-1-one derivatives GLAXO GROUP LIMITED (GB) 1994-11-01 US disclosed