SCHEMBL11020734

SCHEMBL11020734

COc1cc(SC)ccc1-c1nc2ccc(C(=O)O)cc2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 7/20 0.54
PDE4A P27815 5/20 0.52
PDE4B Q07343 5/20 0.52
PDE4C Q08493 5/20 0.52
PDE4D Q08499 5/20 0.52
TDP1 Q9NUW8 3/20 0.52
POLB P06746 3/20 0.52
TP53 P04637 2/20 0.52
MAPT P10636 2/20 0.52
HDAC6 Q9UBN7 1/20 0.49
NR4A2 P43354 1/20 0.48
HSP90AA1 P07900 1/20 0.48
ESR2 Q92731 1/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
F2 P00734 1/20 0.46
F10 P00742 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11020731 0.91 NPC1 (0.44) CHEK2PDE4APDE4BPDE4CPDE4D
SCHEMBL11022051 0.90 CHEK2 (0.66) CHEK2
SCHEMBL11019907 0.90 CHEK2 (0.53) CHEK2MAPTHDAC6HSP90AA1NPC1
SCHEMBL11017274 0.88 CHEK2 (0.56) CHEK2HDAC6HSP90AA1NPC1RAB9A
SCHEMBL11020400 0.88 CHEK2 (0.51) CHEK2PDE4APDE4BPDE4CPDE4D
SCHEMBL11017902 0.88 CHEK2 (0.53) CHEK2PDE4APDE4BPDE4CPDE4D
SCHEMBL20982494 0.86 CHEK2 (0.62) CHEK2PDE4APDE4BPDE4CPDE4D
SCHEMBL11018149 0.86 HDAC6 (0.52) CHEK2POLBHDAC6HSP90AA1NPC1
SCHEMBL11019275 0.85 CHEK2 (0.48) CHEK2PDE4APDE4BPDE4CPDE4D
SCHEMBL3168707 0.82 HDAC6 (0.62) CHEK2PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed