SCHEMBL11022144

SCHEMBL11022144

N#CCC(c1ccccc1)C(Br)Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.50
PBRM1 Q86U86 1/20 0.42
TSHR P16473 2/20 0.40
TAAR1 Q96RJ0 2/20 0.38
HRH1 P35367 4/20 0.37
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
LMNA P02545 1/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
SLC6A2 P23975 2/20 0.35
HTR2A P28223 5/20 0.34
CYP1A2 P05177 2/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CNR1 P21554 1/20 0.33
HKDC1 Q2TB90 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19762907 0.81 TAAR1 (0.55) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL27704927 0.81 TRPA1 (0.48) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL27948315 0.80 TRPA1 (0.52) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL10509394 0.78 TRPA1 (0.41) TRPA1PBRM1TSHRTAAR1HRH1
Water SCHEMBL5164513 0.77 PBRM1 (0.47) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL3952853 0.77 PBRM1 (0.47) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL11565191 0.76 TRPA1 (0.46) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL7007862 0.75 ESR1 (0.47) TRPA1PBRM1TSHRTAAR1HRH1
SCHEMBL28510315 0.72 PBRM1 (0.42) TRPA1PBRM1TSHRTAAR1
SCHEMBL10940254 0.71 PBRM1 (0.43) TRPA1PBRM1TSHRTAAR1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4536599-A HYDROLYZING THE NITRILE DERIVATIVE TO THE AMIDE USING AN ORGANIC QUATERNARY AMINE SALT CATALYST; EFFICIENCY SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1985-08-20 US disclosed
EP-0040896-B1 SYNTHESIS OF AMIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1984-04-25 EP disclosed
EP-0040896-A2 Synthesis of amides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-12-02 EP disclosed
EP-0008532-A1 Synthesis of amines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-03-05 EP disclosed