SCHEMBL11027019

SCHEMBL11027019

COc1ccc(Cc2cc[nH]c(=O)c2C#N)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.47
DAO P14920 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 3/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
BRD4 O60885 2/20 0.40
DHFR P00374 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 2/20 0.38
ATM Q13315 2/20 0.38
GRM2 Q14416 1/20 0.38
KDM4E B2RXH2 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11020707 0.83 PDE3B (0.40) DAOKMT2AGRM2KDM4EHPGD
SCHEMBL11021760 0.81 DAO (0.44) DAOKMT2ADHFRHTTKDM4E
SCHEMBL11021220 0.79 HSD11B1 (0.46) DAOTSHRHTTKDM4EALDH1A1
SCHEMBL11026202 0.76 KDM4E (0.56) DAOKMT2ABRD4POLBKDM4E
SCHEMBL11023987 0.75 DAO (0.42) DAOKMT2APOLBKDM4EALDH1A1
SCHEMBL9356557 0.75 CYP3A4 (0.44) DAOCYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL103159 0.74 MAPT (0.49) CYP3A4CYP2C9KMT2AHTTPOLB
SCHEMBL18796800 0.73 PDE3B (0.68) CA2DAOCYP3A4CYP2C9TSHR
SCHEMBL11021852 0.72 PNP (0.40) CYP3A4TSHRCYP2C19PDE4APDE4B
SCHEMBL11021805 0.71 KDM4E (0.45) DAOKMT2ABRD4POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154190-A1 Pyridones MERCK PATENT GmbH (DE) 1985-09-11 EP disclosed