SCHEMBL11033976

SCHEMBL11033976

Nc1cccc(C(=O)c2cccc(F)c2)c1-c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 3/20 0.47
CDK5R1 Q15078 3/20 0.47
NPC1 O15118 3/20 0.45
RAB9A P51151 2/20 0.45
TACR3 P29371 1/20 0.44
MAPT P10636 2/20 0.43
PARP1 P09874 1/20 0.43
GAA P10253 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
MAPK14 Q16539 1/20 0.43
LMNA P02545 3/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41
GRM5 P41594 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11033978 0.83 CDK5 (0.47) CDK5CDK5R1NPC1RAB9ATACR3
SCHEMBL4416792 0.81 MAPT (0.65) NPC1RAB9AMAPTPARP1GAA
SCHEMBL29963651 0.81 MAPT (0.65) NPC1RAB9AMAPTPARP1GAA
SCHEMBL10372554 0.77 DHODH (0.50) CDK5CDK5R1MAPTCCNA2CDK2
SCHEMBL8586217 0.74 KMT2A (0.66) CDK5CDK5R1NPC1RAB9AMAPT
SCHEMBL4960341 0.73 USP2 (0.52) NPC1RAB9APARP1LMNACES2
SCHEMBL1642906 0.72 KMT2A (0.50) CDK5CDK5R1RAB9AMAPTPARP1
SCHEMBL27883175 0.72 HCRTR1 (0.48) NPC1RAB9ALMNACES2CES1
SCHEMBL1513045 0.72 CES2 (0.57) NPC1RAB9AMAPTPARP1GAA
SCHEMBL15628232 0.71 PARP1 (0.53) CDK5CDK5R1NPC1MAPTPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4518603-A ANTIDEPRESSANTS A. H. ROBINS COMPANY, INC. (US) 1985-05-21 US disclosed