SCHEMBL11041540

SCHEMBL11041540

COc1ccc2c(c1)CC(=S)[N]C=C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
CYP11B1 P15538 6/20 0.41
CYP11B2 P19099 6/20 0.41
BCL2 P10415 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
DRD2 P14416 3/20 0.37
DRD1 P21728 3/20 0.37
DRD5 P21918 3/20 0.37
DRD3 P35462 3/20 0.37
METAP1 P53582 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
DRD4 P21917 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913238 0.81 GAA (0.56) GAACYP11B1CYP11B2BCL2MAOA
SCHEMBL11129395 0.75 GAA (0.49) GAACYP11B1CYP11B2BCL2MAOA
Hydrochloric Acid SCHEMBL11039966 0.74 GAA (0.48) GAACYP11B1CYP11B2BCL2MAOA
SCHEMBL11044464 0.72 GAA (0.68) GAACYP11B1CYP11B2BCL2MAOA
SCHEMBL322514 0.71 TRPA1 (0.39) GAACYP11B1CYP11B2CYP1A2CA1
SCHEMBL1091043 0.67 CA12 (0.39) CYP1A2CA1CA2
SCHEMBL4133299 0.67 GAA (0.50) GAACYP11B1CYP11B2BCL2MAOA
SCHEMBL31463289 0.67 GAA (0.50) GAACYP11B1CYP11B2BCL2MAOA
SCHEMBL10232028 0.67 GAA (0.57) GAACYP11B1CYP11B2BCL2MAOA
SCHEMBL14181700 0.66 CYP11B1 (0.54) GAACYP11B1CYP11B2BCL2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP disclosed