SCHEMBL11041853

SCHEMBL11041853

O=C1NC(=O)C(c2cccc3ccc(F)cc23)O1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.56
CA2 P00918 2/20 0.43
GSK3B P49841 3/20 0.41
ADK P55263 2/20 0.41
PTGER3 P43115 4/20 0.39
TYMS P04818 2/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
PRKDC P78527 1/20 0.35
CYP1B1 Q16678 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPK1 P28482 2/20 0.35
LMNA P02545 1/20 0.35
TDP2 O95551 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
ALOX12 P18054 1/20 0.34
CASP3 P42574 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11043656 0.83 CA2 (0.43) IDO1CA2PTGER3TYMSKDM4E
SCHEMBL11039068 0.82 CA2 (0.54) IDO1CA2GSK3BADKKDM4E
SCHEMBL11040694 0.74 CA2 (0.47) CA2KDM4EALDH1A1LMNAMAPT
SCHEMBL11040723 0.73 CA2 (0.64) CA2KDM4E
SCHEMBL11041002 0.72 CA2 (0.58) CA2KDM4EALDH1A1LMNA
SCHEMBL17258148 0.72 IDO1 (1.00) IDO1LMNAMAPTCYP2C19ABCG2
SCHEMBL11047713 0.71 CA2 (0.49) CA2PTGER3CYP1A1CYP1A2CYP1B1
SCHEMBL10545336 0.71 CA2 (0.42) CA2CASP3BLMSENP8SENP7
SCHEMBL11041960 0.70 CA2 (0.60) CA2
SCHEMBL11040315 0.69 CA2 (0.67) CA2GSK3BNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448971-A Hypoglycemic 5-phenyl-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1984-05-15 US disclosed
US-4407811-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1983-10-04 US disclosed
US-4399296-A TRIMETHYLSILYL CYANOHYDRIN INTERMEDIATES PFIZER INC. (US) 1983-08-16 US disclosed
US-4367234-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1983-01-04 US disclosed