SCHEMBL11042441

SCHEMBL11042441

COc1ccc(C(=O)N2CCN(C(=O)c3ccc4c(c3)CCC(=O)N4)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.66
PGR P06401 1/20 0.66
SLC6A4 P31645 1/20 0.66
KCNH2 Q12809 1/20 0.66
PDE3B Q13370 1/20 0.66
PDE3A Q14432 1/20 0.66
CRBN Q96SW2 6/20 0.54
HPGD P15428 1/20 0.53
ALDH1A1 P00352 3/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
GLA P06280 1/20 0.51
ALOX15 P16050 1/20 0.51
MAPK1 P28482 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
DRD2 P14416 4/20 0.50
DRD3 P35462 2/20 0.50
PKM P14618 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060430 0.90 NR3C1 (0.58) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11202820 0.90 NR3C1 (0.78) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11045173 0.90 NR3C1 (0.57) NR3C1PGRSLC6A4KCNH2PDE3B
Hydrochloric Acid SCHEMBL11042554 0.90 NR3C1 (0.57) NR3C1PGRSLC6A4KCNH2PDE3B
Hydrochloric Acid SCHEMBL11039493 0.90 NR3C1 (0.57) NR3C1PGRSLC6A4KCNH2PDE3B
Water SCHEMBL11200345 0.89 NR3C1 (0.76) NR3C1PGRSLC6A4KCNH2PDE3B
Water SCHEMBL11200349 0.89 NR3C1 (0.76) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL7325459 0.89 NR3C1 (0.56) NR3C1PGRSLC6A4KCNH2PDE3B
Hydrochloric Acid SCHEMBL7350304 0.89 NR3C1 (0.54) NR3C1PGRSLC6A4KCNH2PDE3B
Hydrochloric Acid SCHEMBL11042650 0.88 DRD3 (0.66) NR3C1PGRSLC6A4KCNH2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed