SCHEMBL11047794

SCHEMBL11047794

COC(c1c[nH]cn1)c1ccccc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.46
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
ADRA2A P08913 4/20 0.34
ADRA2B P18089 4/20 0.34
ADRA2C P18825 3/20 0.34
CYP2D6 P10635 2/20 0.33
SLC22A2 O15244 1/20 0.33
SLC22A1 O15245 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
DRD1 P21728 1/20 0.33
HRH2 P25021 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11051380 0.84 ESR1 (0.42) ESR1SLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL11047824 0.83
SCHEMBL10552827 0.80 ESR1 (0.38) ESR1SLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL2105209 0.79 ADRA2A (0.38) ESR1SLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL11047860 0.79 ESR1 (0.37) ESR1SLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL6210930 0.76 ADRA2A (0.36) ADRA2AADRA2BADRA2CCYP2D6CYP2C19
SCHEMBL23109096 0.76 ESR1 (0.50) ESR1SLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL8027681 0.75 CYP19A1 (0.37) ESR1SLC6A2SLC6A4SLC6A3ADRA2A
Hydrochloric Acid SCHEMBL6218208 0.75 ADRA2A (0.37) ADRA2AADRA2BADRA2CCYP2D6CYP2C19
SCHEMBL13089136 0.73 MAPT (0.42) ESR1SLC6A2SLC6A4SLC6A3ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4443466-A DIURETICS, SEDATIVES, ANALGESICS Farmos-Yhtyma OY (Farmos Group Ltd.) (FI) 1984-04-17 US claimed
EP-0024829-B1 4-BENZYL- AND 4-BENZOYLIMIDAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Farmos-Yhtyma Oy (FI) 1984-04-25 EP disclosed
US-4443466-A DIURETICS, SEDATIVES, ANALGESICS Farmos-Yhtyma OY (Farmos Group Ltd.) (FI) 1984-04-17 US disclosed