SCHEMBL11049503

SCHEMBL11049503

CC(C)(C)NC(=O)NC(=N)Nc1ccc(Br)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.71
RAB9A P51151 6/20 0.71
MEN1 O00255 5/20 0.71
NPC1 O15118 5/20 0.71
HTT P42858 3/20 0.53
SMN1; SMN2 Q16637 4/20 0.48
LMNA P02545 4/20 0.48
POLB P06746 1/20 0.48
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
FPR2 P25090 1/20 0.45
MAPT P10636 3/20 0.44
EPHX1 P07099 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPK1 P28482 1/20 0.43
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052142 0.86 MEN1 (0.53) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11052517 0.85 NPC1 (0.50) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11054637 0.84 HTT (0.52) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11049538 0.84 NPC1 (0.49) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11056203 0.84 NPC1 (0.49) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11060416 0.82 GAA (0.49) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11052448 0.82 EPHX2 (0.56) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11249625 0.81 HTT (0.53) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL11244605 0.81 HTT (0.50) KMT2ARAB9AMEN1NPC1HTT
SCHEMBL10756539 0.81 MDM2 (0.50) KMT2ARAB9AMEN1NPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed