SCHEMBL11060416

SCHEMBL11060416

CC(C)(C)NC(=O)NC(=N)Nc1cccc(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
RAB9A P51151 4/20 0.48
NPC1 O15118 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TGM2 P21980 1/20 0.46
TRPV1 Q8NER1 1/20 0.45
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 1/20 0.44
GRIK1 P39086 2/20 0.43
GRIK2 Q13002 2/20 0.43
P2RX1 P51575 1/20 0.43
MAPK1 P28482 1/20 0.42
STING1 Q86WV6 1/20 0.42
ANO1 Q5XXA6 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056203 0.85 NPC1 (0.49) GAARAB9ANPC1MEN1KMT2A
SCHEMBL21928147 0.85 RAB9A (0.65) GAARAB9ANPC1MEN1KMT2A
SCHEMBL11050011 0.84 MEN1 (0.50) GAARAB9ANPC1MEN1KMT2A
SCHEMBL11053687 0.83 MEN1 (0.55) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL11052517 0.83 NPC1 (0.50) GAARAB9ANPC1MEN1KMT2A
SCHEMBL11049503 0.82 KMT2A (0.71) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL11056636 0.81 SMN1; SMN2 (0.59) GAARAB9AMEN1KMT2ATRPV1
SCHEMBL17777456 0.80 MEN1 (0.55) GAARAB9ANPC1MEN1KMT2A
SCHEMBL11249625 0.80 HTT (0.53) GAARAB9ANPC1MEN1KMT2A
SCHEMBL11244605 0.80 HTT (0.50) GAARAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed