SCHEMBL11049547

SCHEMBL11049547

[O-][S+]1CCN(c2nc(NCCCCCO)nc3c(SCc4ccccc4)ncnc23)CC1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 13/20 0.40
CYP1A2 P05177 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
PPARG P37231 3/20 0.37
KCNH3 Q9ULD8 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
NCOA2 Q15596 1/20 0.36
PDGFRA P16234 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10972196 1.00 SLC29A1 (0.40) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL11046570 0.96 CYP1A2 (0.40) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL2460092 0.93 SLC29A1 (0.45) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL11052740 0.89 KCNH3 (0.39) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL11026335 0.89 PDE4A (0.44) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL10970925 0.89 SLC29A1 (0.43) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL10971507 0.86 CYP1A2 (0.37) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL11029641 0.85 PDE4A (0.42) SLC29A1CYP1A2PDE4APDE4BPDE4C
SCHEMBL11047084 0.85 PDE4A (0.41) SLC29A1PDE4APDE4BPDE4CPDE4D
SCHEMBL11031378 0.85 RCE1 (0.36) SLC29A1CYP1A2PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478833-A ANTICOAGULANTS DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-10-23 US disclosed
EP-0055444-A2 Trisubstituted pyrimido(5,4-d)pyrimidines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-07-07 EP disclosed