SCHEMBL11050475

SCHEMBL11050475

CC(C)(C)NC(=O)NC(=N)Nc1cc(Br)ccc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
NPC1 O15118 5/20 0.48
RAB9A P51151 5/20 0.48
MAPK1 P28482 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
LMNA P02545 4/20 0.42
GAA P10253 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
THRB P10828 1/20 0.42
BLM P54132 1/20 0.42
BTK Q06187 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PLK3 Q9H4B4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11050905 0.89 NPC1 (0.51) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11258056 0.88 MEN1 (0.47) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11053819 0.86 KMT2A (0.46) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11051067 0.86 HTT (0.43) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11055583 0.85 MAPT (0.47) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11053662 0.84 NPC1 (0.49) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11048661 0.84 MAPK1 (0.52) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11056245 0.84 NPC1 (0.46) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2
SCHEMBL11051039 0.83 HTT (0.49) ALDH1A1NPC1RAB9AMAPK1MEN1
SCHEMBL11053893 0.82 RAB9A (0.43) ALDH1A1NPC1RAB9AMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed