SCHEMBL11053451

SCHEMBL11053451

COc1ccc2c(c1)CC1CCC(C2)C1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.61
DRD3 P35462 6/20 0.61
PSEN1 P49768 1/20 0.48
PSEN2 P49810 1/20 0.48
APH1B Q8WW43 1/20 0.48
NCSTN Q92542 1/20 0.48
APH1A Q96BI3 1/20 0.48
PSENEN Q9NZ42 1/20 0.48
CYP19A1 P11511 3/20 0.47
DRD4 P21917 2/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
KDM1A O60341 1/20 0.43
CA2 P00918 3/20 0.43
CA1 P00915 2/20 0.43
ACHE P22303 2/20 0.43
CYP26A1 O43174 1/20 0.43
KYAT1 Q16773 1/20 0.42
KYAT3 Q6YP21 1/20 0.42
AADAT Q8N5Z0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11222319 0.98 DRD2 (0.59) DRD2DRD3PSEN1PSEN2APH1B
SCHEMBL295336 0.82 DRD2 (0.74) DRD2DRD3CYP19A1DRD4MTNR1A
SCHEMBL20542100 0.82 DRD2 (0.74) DRD2DRD3CYP19A1DRD4MTNR1A
SCHEMBL20541972 0.82 DRD2 (0.74) DRD2DRD3CYP19A1DRD4MTNR1A
SCHEMBL30579427 0.82 DRD2 (0.74) DRD2DRD3CYP19A1DRD4MTNR1A
Hydrochloric Acid SCHEMBL1788371 0.80 DRD2 (0.72) DRD2DRD3CYP19A1DRD4MTNR1A
SCHEMBL11047950 0.76 DRD2 (0.43) DRD2DRD3PSEN1PSEN2APH1B
SCHEMBL11055734 0.76 METAP1 (0.50) DRD2DRD3CYP19A1ACHECYP26A1
SCHEMBL267102 0.76 DRD2 (1.00) DRD2DRD3CYP19A1DRD4MTNR1A
SCHEMBL354006 0.76 DRD2 (1.00) DRD2DRD3CYP19A1DRD4MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4454325-A ANALGESICS MERCK SHARP & DOHME I.A. CORP. (US) 1984-06-12 US disclosed
US-4376779-A N-(Substituted)-2-aza-2'-hydroxy-5,6-benzotricyclo[6.3.01,8.04,11 ] undecane centrally-acting analgesics MERCK SHARP & DOHME (I.A.) CORP. (US) 1983-03-15 US disclosed