SCHEMBL11063231

SCHEMBL11063231

CC(C)NC(=O)C(C)N1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.54
CHRM5 P08912 1/20 0.51
CHRM3 P20309 1/20 0.51
CYP1A2 P05177 2/20 0.44
PABPC1 P11940 1/20 0.41
APOBEC3A P31941 1/20 0.41
EIF4H Q15056 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
ATM Q13315 2/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CA2 P00918 1/20 0.35
CHKA P35790 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.34
OPRD1 P41143 2/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5485542 0.98 SIGMAR1 (0.52) SIGMAR1CHRM5CHRM3CYP1A2PABPC1
SCHEMBL23835774 0.84 ATM (0.50) SIGMAR1PABPC1APOBEC3AEIF4HAPOBEC3G
SCHEMBL11064005 0.82 SIGMAR1 (0.51) SIGMAR1CHRM5CHRM3CYP1A2ATM
SCHEMBL11066704 0.82 SIGMAR1 (0.49) SIGMAR1CHRM5CHRM3CYP1A2KDM4E
SCHEMBL27536506 0.79 SIGMAR1 (0.46) SIGMAR1CHRM5CHRM3CYP1A2MEN1
SCHEMBL24069101 0.79 CHRM5 (0.46) SIGMAR1CHRM5CHRM3CYP1A2CA2
SCHEMBL23866564 0.78 KDM4E (0.55) SIGMAR1CYP1A2PABPC1APOBEC3AEIF4H
SCHEMBL23866568 0.78 KDM4E (0.55) SIGMAR1CYP1A2PABPC1APOBEC3AEIF4H
SCHEMBL21661626 0.78 KDM4E (0.55) SIGMAR1CYP1A2PABPC1APOBEC3AEIF4H
SCHEMBL6678936 0.78 SIGMAR1 (0.58) SIGMAR1CHRM5CHRM3KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478838-A VASODILATOR AGENTS HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1984-10-23 US disclosed
EP-0083712-A1 1-(3,4,5-Trimethoxycinnamoyl)-4-aminocarbonylethyl-substituted piperazine derivatives and a process for the preparation thereof Hokuriku Pharmaceutical Co.,Ltd (JP) 1983-07-20 EP disclosed