SCHEMBL11065170

SCHEMBL11065170

CNC(=O)Nc1ccc(-c2ccncc2)c(C)n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 13/20 0.47
ADORA2A P29274 9/20 0.47
ADORA1 P30542 8/20 0.47
ABL1 P00519 1/20 0.45
GCK P35557 1/20 0.45
ADORA3 P0DMS8 4/20 0.44
CYP46A1 Q9Y6A2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11069813 0.85 ADORA2B (0.44) ADORA2BADORA2AADORA1ABL1ADORA3
SCHEMBL11065275 0.83 ADORA2B (0.45) ADORA2BADORA2AADORA1ABL1GCK
SCHEMBL11066718 0.81 ADORA2B (0.44) ADORA2BADORA2AADORA1ABL1GCK
SCHEMBL11069532 0.80 SMN1; SMN2 (0.51) ADORA2BADORA2AADORA1ADORA3ALDH1A1
SCHEMBL11069278 0.80 ADORA2B (0.43) ADORA2BADORA2AADORA1ABL1GCK
SCHEMBL11071690 0.79 ADORA2B (0.42) ADORA2BADORA2AADORA1ABL1GCK
SCHEMBL11070623 0.79 ADORA2B (0.42) ADORA2BADORA2AADORA1ABL1GCK
SCHEMBL11694093 0.75 POLB (0.64) ABL1GCKALDH1A1POLB
SCHEMBL11063569 0.74 PDE3B (0.42) ADORA2BADORA2AADORA1ADORA3CYP46A1
SCHEMBL7056328 0.72 CDK5 (0.68) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448780-A N-(Lower-alkyl)-N'-[5-(pyridinyl)-2-pyridinyl]ureas and cardiotonic use thereof STERLING DRUG INC. (US) 1984-05-15 US claimed
US-4448780-A N-(Lower-alkyl)-N'-[5-(pyridinyl)-2-pyridinyl]ureas and cardiotonic use thereof STERLING DRUG INC. (US) 1984-05-15 US disclosed