SCHEMBL11065308

SCHEMBL11065308

CCC1C(=O)C(C)CC(C(=O)OC)C1=O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CYP1A2 P05177 1/20 0.33
HIF1A Q16665 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 1/20 0.31
GAA P10253 2/20 0.31
LMNA P02545 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11062852 0.89 TSHR (0.34) CYP1A2HIF1AALDH1A1LMNA
SCHEMBL11069510 0.80 CYP1A2 (0.35) BRD4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL11059934 0.79 TSHR (0.33) BRD4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL11055929 0.75 BRD4 (0.33) BRD4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL11062454 0.75 CYP1A2 (0.35) BRD4CYP1A2HIF1AALDH1A1
SCHEMBL11061482 0.74 TSHR (0.33) BRD4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL11059896 0.72 ALDH1A1 (0.36) BRD4CYP1A2HIF1AALDH1A1GAA
SCHEMBL5896869 0.71 ALDH1A1 (0.39) BRD4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL11062133 0.69 ALDH1A1 (0.34) BRD4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL11061512 0.69 ALDH1A1 (0.32) CYP1A2HIF1AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4432378-A ORGANOLEPTIC; TOBACCO; FOODS; DETERGENTS; COSMETICS FRITZSCHE, DODGE & OLCOTT, INC. (US) 1984-02-21 US disclosed
US-4326996-A FOR PERFUMES FRITZSCHE DODGE & OLCOTT INC. (US) 1982-04-27 US disclosed
US-4281204-A ALKYLATION, DECARBOXYLATION TO CYCLIZE FRITZSCHE DODGE & OLCOTT INC. (US) 1981-07-28 US disclosed