SCHEMBL11068634

SCHEMBL11068634

CC1CC(NC(=O)C(F)(F)F)=NN1c1ccc(-c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.47
GAA P10253 2/20 0.47
MEN1 O00255 8/20 0.41
KMT2A Q03164 8/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
TP53 P04637 2/20 0.41
HSD17B10 Q99714 1/20 0.41
ATM Q13315 3/20 0.38
CACNA1H O95180 1/20 0.38
CACNA1C Q13936 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
ACHE P22303 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MAPT P10636 3/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11061030 0.86 ABL1 (0.50) ABL1GAAMEN1KMT2ACACNA1H
SCHEMBL11061324 0.85 ABL1 (0.55) ABL1GAAMEN1KMT2ANPC1
SCHEMBL11060498 0.84 ABL1 (0.48) ABL1GAAHDAC6PDE5A
SCHEMBL11054662 0.80 ABL1 (0.74) ABL1GAAPDE5A
SCHEMBL11057356 0.79 GAA (0.55) GAAMEN1KMT2AATML3MBTL1
SCHEMBL11059709 0.77 NR3C2 (0.49) GAAMEN1KMT2AATMCACNA1H
SCHEMBL10657219 0.77 ABL1 (0.66) ABL1GAAMEN1KMT2ANPC1
SCHEMBL11063665 0.76 MEN1 (0.49) GAAMEN1KMT2AATML3MBTL1
SCHEMBL11060638 0.75 PDE5A (0.50) GAAMEN1KMT2AATML3MBTL1
SCHEMBL11058352 0.74 ABL1 (0.49) ABL1GAAMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447442-A ANTIINFLAMMATORY, ANTIARTHRITIC, ANTIHISTAMINE, ANTIALLERGENS, ANALGESICS, BACTERICIDES, AND FUNGICIDES AMERICAN CYANAMID COMPANY (US) 1984-05-08 US disclosed
EP-0070376-A1 Heterocyclic substituted-amino-pyrazolines AMERICAN CYANAMID COMPANY (US) 1983-01-26 EP disclosed
US-4348527-A ANALGESICS, BACTERICIDES, FUNGICIDES AMERICAN CYANAMID COMPANY (US) 1982-09-07 US disclosed