SCHEMBL11070880

SCHEMBL11070880

CCCCCCCCN1C2=NCCN2C(=O)c2nc(C(C)C)[nH]c21

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 1/20 0.38
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
LMNA P02545 2/20 0.32
TSHR P16473 2/20 0.32
HTT P42858 1/20 0.32
PTGS1 P23219 3/20 0.31
PTGS2 P35354 3/20 0.31
MGLL Q99685 2/20 0.31
FAAH O00519 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
PNP P00491 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11067126 0.85 MEN1 (0.46) MEN1KMT2AALDH1A1PDE3BPDE3A
SCHEMBL11070883 0.83 MEN1 (0.44) MEN1KMT2AALDH1A1PDE3BPDE3A
SCHEMBL10800120 0.76 MEN1 (0.49) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL11074233 0.66 PDE4A (0.45) MEN1KMT2AALDH1A1CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL10795748 0.65 MEN1 (0.47) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL11802972 0.65 MEN1 (0.54) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL10798493 0.63 TSHR (0.54) MEN1KMT2ACYP2D6LMNATSHR
SCHEMBL9585449 0.58 PDE4A (0.44) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL7153652 0.56 MGLL (0.60) ALDH1A1PTGS1PTGS2MGLLFAAH
SCHEMBL17999908 0.54 MGLL (0.64) ALDH1A1LMNATSHRHTTPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US claimed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US claimed