SCHEMBL11072066

SCHEMBL11072066

CCCCn1c(=S)c2[nH]cnc2n(CCCC)c1=O

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 15/20 0.70
PDE4B Q07343 15/20 0.70
PDE4C Q08493 15/20 0.70
PDE4D Q08499 15/20 0.70
ADORA2A P29274 11/20 0.70
ADORA2B P29275 8/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080222 0.99 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11153561 0.96 ADORA2B (0.76) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7094603 0.92 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11489193 0.87 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3186630 0.85 PDE4A (0.94) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11361392 0.84 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3190853 0.82 ADORA2B (0.92) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381259 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381240 0.82 ADORA2B (0.94) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3842077 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4454138-A TREATMENT OF VASCULAR DISEASES Wuelfing, Johann A. (DE) 1984-06-12 US disclosed
EP-0018136-B1 XANTHINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS BEECHAM - WUELFING GmbH & Co. KG (DE) 1983-11-16 EP disclosed
EP-0018136-A1 Xanthine derivatives, a process for their preparation and their use in pharmaceutical compositions BEECHAM - WUELFING GmbH & Co. KG (DE) 1980-10-29 EP disclosed