SCHEMBL11073096

SCHEMBL11073096

CCCCCC1CCc2cc(C(N)=O)ccc2C1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.57
CYP2C8 P10632 2/20 0.57
S1PR3 Q99500 2/20 0.57
CYP2C9 P11712 2/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C19 P33261 1/20 0.57
S1PR1 P21453 7/20 0.48
SGPL1 O95470 3/20 0.48
S1PR4 O95977 1/20 0.48
S1PR5 Q9H228 1/20 0.48
DRD3 P35462 4/20 0.47
ITGB3 P05106 2/20 0.42
ITGA2B P08514 2/20 0.42
DRD2 P14416 2/20 0.41
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11215122 0.99 CYP3A4 (0.59) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11209578 0.95 CYP3A4 (0.52) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11214160 0.94 CYP3A4 (0.54) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11072230 0.88 CYP3A4 (0.56) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11074273 0.88 CYP3A4 (0.58) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL8553934 0.88 CYP3A4 (0.46) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11209754 0.87 CYP3A4 (0.57) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL12065071 0.84 CYP3A4 (0.54) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11063644 0.83 CYP3A4 (0.53) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6
SCHEMBL11072113 0.83 CYP3A4 (0.50) CYP3A4CYP2C8S1PR3CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4462923-A Disubstituted pyrimidines HOFFMANN-LA ROCHE INC. (US) 1984-07-31 US disclosed
US-4391731-A Hydrogenated naphthalenes HOFFMANN-LA ROCHE INC. (US) 1983-07-05 US disclosed
EP-0047817-A2 Hydrogenated naphthalines, their preparation and application, and mixtures containing such naphthalines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-03-24 EP disclosed