SCHEMBL11075149

SCHEMBL11075149

COc1cccc(C23CC2C(=O)NC3=O)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.50
KDM1A O60341 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
SIGMAR1 Q99720 2/20 0.43
DDB1 Q16531 2/20 0.43
CRBN Q96SW2 2/20 0.43
CXCR3 P49682 1/20 0.43
ADAM17 P78536 1/20 0.42
CTSD P07339 1/20 0.42
CTSE P14091 1/20 0.42
BACE1 P56817 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11761376 0.83 MEN1 (0.41) KDM1AMEN1KMT2APOLBSMN1; SMN2
SCHEMBL11911732 0.82 CYP19A1 (0.64) CYP19A1DDB1CRBNCXCR3CTSE
SCHEMBL12313146 0.82 CYP19A1 (0.64) CYP19A1DDB1CRBNCXCR3CTSE
SCHEMBL11075680 0.82 CYP19A1 (0.64) CYP19A1DDB1CRBNCXCR3CTSE
SCHEMBL11085029 0.78 CYP19A1 (0.54) CYP19A1KDM1A
SCHEMBL10533819 0.78 CYP19A1 (0.67) CYP19A1DDB1CRBNCXCR3BACE1
SCHEMBL11088395 0.78 CYP19A1 (0.54) CYP19A1KDM1AMEN1KMT2ADDB1
SCHEMBL1552771 0.76 CYP19A1 (0.69) CYP19A1KDM1AMEN1KMT2APOLB
SCHEMBL2054565 0.76 CYP19A1 (0.69) CYP19A1KDM1AMEN1KMT2APOLB
SCHEMBL15196027 0.76 CYP19A1 (0.69) CYP19A1KDM1AMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4435419-A Method of treating depression using azabicyclohexanes AMERICAN CYANAMID COMPANY (US) 1984-03-06 US disclosed
US-4231935-A ANXIOLYTICS AND ANALGESICS AMERICAN CYANAMID COMPANY (US) 1980-11-04 US disclosed
US-4196120-A 1,2-BIS(HYDROCARBYLSULFONYLOXY OR HALO METHYL)CYCLOPROPYLBENZENE, OPTICAL ACITIVITY ANALGESICS AMERICAN CYANAMID COMPANY (US) 1980-04-01 US disclosed
US-4131611-A ANXIOLYTIC, ANALGESIC AMERICAN CYANAMID COMPANY (US) 1978-12-26 US disclosed