SCHEMBL11075196

SCHEMBL11075196

N#Cc1cc2c([nH]c1=O)oc1ncccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 4/20 0.39
LRRK2 Q5S007 1/20 0.39
HPGD P15428 3/20 0.37
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
LMNA P02545 2/20 0.37
PDE5A O76074 1/20 0.37
TSHR P16473 1/20 0.37
PTGS1 P23219 1/20 0.37
PDE4A P27815 1/20 0.37
CYP2C19 P33261 1/20 0.37
BLM P54132 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
CDK5 Q00535 2/20 0.36
CDK5R1 Q15078 2/20 0.36
CLK1 P49759 1/20 0.36
CLK2 P49760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11068415 0.80 KDM4E (0.44) KDM4EALDH1A1LRRK2HPGDPDE3B
SCHEMBL11069631 0.77 KDM4E (0.48) KDM4EALDH1A1HPGDLMNAGALR3
SCHEMBL11071799 0.74 ALDH1A1 (0.38) KDM4EALDH1A1PARP1AURKA
SCHEMBL11071485 0.73 LRRK2 (0.39) KDM4EALDH1A1LRRK2HPGDPDE3B
SCHEMBL11071409 0.73 PDE3B (0.43) KDM4EHPGDPDE3BPDE3ALMNA
SCHEMBL11071637 0.73 PDE3B (0.43) KDM4EALDH1A1HPGDPDE3BPDE3A
SCHEMBL7338498 0.71 PARP1 (0.47) KDM4ELRRK2HPGDPDE3BPDE3A
SCHEMBL7339417 0.69 PARP1 (0.47) KDM4EALDH1A1HPGDPDE3BPDE3A
SCHEMBL30421743 0.68 DAO (0.59) KDM4EALDH1A1LRRK2HPGDPDE3B
SCHEMBL10689557 0.68 DAO (0.59) KDM4EALDH1A1LRRK2HPGDPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4474786-A CONGESTIVE HEART FAILURE SCHERING CORPORATION (US) 1984-10-02 US disclosed
EP-0102046-A1 Tricyclic lactams, method for making them, pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-03-07 EP disclosed