SCHEMBL11076513

SCHEMBL11076513

CCOc1ccc(C(CN)CNC)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.47
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ADRA2A P08913 2/20 0.41
PLK1 P53350 1/20 0.40
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PARP10 Q53GL7 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
ACACB O00763 2/20 0.38
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11088390 0.87 SLC2A1 (0.47) TSHRSMN1; SMN2CA12CA1CA2
SCHEMBL11080189 0.87 PLK1 (0.43) PLK1ALDH1A1SMN1; SMN2CA12CA1
SCHEMBL11081839 0.86 NQO1 (0.58) NQO1TSHRTDP1ADRA2AALDH1A1
SCHEMBL11070462 0.83 AOC3 (0.49) ALDH1A1CA12CA1CA2CA7
SCHEMBL11069017 0.81 CYP3A4 (0.46) TSHRALDH1A1
SCHEMBL11080230 0.80 MAOB (0.50) SMN1; SMN2LTA4HL3MBTL1MAPT
SCHEMBL11079411 0.77 TDP1 (0.41) TSHRTDP1ADRA2APLK1ALDH1A1
SCHEMBL11074337 0.77 CYP2D6 (0.39) TSHRTDP1ALDH1A1SMN1; SMN2NPSR1
SCHEMBL11084756 0.77 TAAR1 (0.37) TSHRTDP1ADRA2AALDH1A1SMN1; SMN2
SCHEMBL11073428 0.75 GABBR2 (0.50) TDP1ADRA2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed