SCHEMBL11077085

SCHEMBL11077085

COc1ccc(-n2ccnc2)c([N+](=O)[O-])c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
MAPK1 P28482 1/20 0.57
GRIK1 P39086 1/20 0.52
GRIA1 P42261 1/20 0.52
GRIA2 P42262 1/20 0.52
GRIA3 P42263 1/20 0.52
GRIA4 P48058 1/20 0.52
GRIK2 Q13002 1/20 0.52
GRIK3 Q13003 1/20 0.52
GRIK4 Q16099 1/20 0.52
GRIK5 Q16478 1/20 0.52
CYP11B1 P15538 2/20 0.51
CYP11B2 P19099 2/20 0.51
MAPT P10636 2/20 0.50
KMT2A Q03164 1/20 0.47
CYP19A1 P11511 1/20 0.47
POLB P06746 1/20 0.46
RECQL P46063 1/20 0.46
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3497031 0.83 GRIK1 (0.49) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL995544 0.82 GRIK1 (0.56) ALDH1A1GRIK1GRIA1GRIA2GRIA3
SCHEMBL11830513 0.81 ALDH1A1 (0.64) ALDH1A1MAPK1GRIK1GRIA1GRIA2
SCHEMBL10786918 0.80 GRIK1 (0.57) ALDH1A1GRIK1GRIA1GRIA2GRIA3
SCHEMBL9692480 0.80 MAPT (0.72) ALDH1A1GRIK1GRIA1GRIA2GRIA3
SCHEMBL29758064 0.79 GRIK1 (0.56) ALDH1A1MAPK1GRIK1GRIA1GRIA2
SCHEMBL28850718 0.79 GRIA1 (0.56) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL1237406 0.79 GRIA1 (0.56) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL11077376 0.79 GRIK1 (0.56) ALDH1A1MAPK1GRIK1GRIA1GRIA2
SCHEMBL10066486 0.78 GRIK1 (0.52) ALDH1A1GRIK1GRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0003560-B1 IMIDAZOLE DERIVATIVES AND SALTS THEREOF, THEIR SYNTHESIS, AND PHARMACEUTICAL FORMULATIONS THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-02 EP disclosed
US-4431815-A CARDIOTONIC AND ANTISHOCK AGENTS; ANTICOAGULANTS BURROUGHS WELLCOME CO. (US) 1984-02-14 US disclosed
EP-0003560-A2 Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations THE WELLCOME FOUNDATION LIMITED (GB) 1979-08-22 EP disclosed