SCHEMBL11078987

SCHEMBL11078987

Clc1ccc(/C=C/Cn2ccnc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 4/20 0.65
CYP2A6 P11509 1/20 0.56
CYP19A1 P11511 1/20 0.56
CYP11B1 P15538 1/20 0.56
CYP11B2 P19099 1/20 0.56
CYP2B6 P20813 1/20 0.56
TP53 P04637 2/20 0.48
KDM4E B2RXH2 1/20 0.48
TSHR P16473 1/20 0.48
CYP1A2 P05177 2/20 0.47
USP2 O75604 1/20 0.47
LMNA P02545 1/20 0.47
MEN1 O00255 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11078989 1.00 TBXAS1 (0.65) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL11148664 0.92 TBXAS1 (0.56) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL11397028 0.92 TBXAS1 (0.56) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL11442580 0.90 TBXAS1 (0.57) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL11379570 0.86 TP53 (0.52) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL8347428 0.83 TBXAS1 (0.68) TBXAS1CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL8347430 0.83 TBXAS1 (0.68) TBXAS1CYP19A1CYP11B1CYP11B2CYP1A2
Hydrochloric Acid SCHEMBL28253387 0.82 TBXAS1 (0.69) TBXAS1CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL11382258 0.81 ITGAL (0.51) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL11146930 0.81 TBXAS1 (0.49) TBXAS1KDM4ETSHRCYP1A2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4396771-A THROMBOEMBOLIC DISORDERS, SHOCK BURROUGHS WELLCOME CO. (US) 1983-08-02 US claimed
US-4431815-A CARDIOTONIC AND ANTISHOCK AGENTS; ANTICOAGULANTS BURROUGHS WELLCOME CO. (US) 1984-02-14 US disclosed
US-4425354-A CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1984-01-10 US disclosed
EP-0003732-B1 IMIDAZOLE DERIVATIVES AND SALTS THEREOF, THEIR SYNTHESIS, AND PHARMACEUTICAL FORMULATIONS THEREOF THE WELLCOME FOUNDATION LIMITED (GB) 1983-10-19 EP disclosed
US-4405634-A Imidazole derivatives for treating myocardial infarction BURROUGHS WELLCOME CO. (US) 1983-09-20 US disclosed
US-4396771-A THROMBOEMBOLIC DISORDERS, SHOCK BURROUGHS WELLCOME CO. (US) 1983-08-02 US disclosed
US-4357340-A Imidazole derivatives and angina pectoris BURROUGHS WELLCOME CO. (US) 1982-11-02 US disclosed
EP-0003732-A2 Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations thereof THE WELLCOME FOUNDATION LIMITED (GB) 1979-09-05 EP disclosed