SCHEMBL11080697

SCHEMBL11080697

CNCC(CN)c1cccc(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 3/20 0.54
KDM4E B2RXH2 1/20 0.49
MTNR1A P48039 2/20 0.47
MTNR1B P49286 2/20 0.47
SLC6A2 P23975 4/20 0.46
SLC6A4 P31645 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CASR P41180 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KCNH2 Q12809 1/20 0.43
CHEK1 O14757 1/20 0.43
ROCK2 O75116 1/20 0.43
RPS6KA5 O75582 1/20 0.43
MAP4K4 O95819 1/20 0.43
CHEK2 O96017 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11081355 0.87 AOC3 (0.54) AOC3MTNR1AMTNR1BL3MBTL1CASR
SCHEMBL28978068 0.86 AOC3 (0.51) AOC3KDM4EMTNR1AMTNR1BSLC6A2
SCHEMBL11083337 0.85 KDM4E (0.43) AOC3KDM4EMTNR1AMTNR1BSLC6A2
SCHEMBL11069017 0.85 CYP3A4 (0.46) AOC3KDM4ESLC6A2SLC6A4CYP3A4
SCHEMBL11085320 0.82 KDM4E (0.42) KDM4EROCK2PRKACARPS6KB1CDK2
SCHEMBL5778033 0.82 AOC3 (0.50) AOC3MTNR1AMTNR1BL3MBTL1CASR
SCHEMBL11081698 0.80 BCHE (0.53) SLC6A2SLC6A4CYP3A4CYP2D6SLC6A3
SCHEMBL11070462 0.80 AOC3 (0.49) AOC3SLC6A2SLC6A4L3MBTL1CYP3A4
SCHEMBL7411654 0.79 AOC3 (0.48) AOC3MTNR1AMTNR1BL3MBTL1CASR
SCHEMBL7376528 0.79 AOC3 (0.48) AOC3MTNR1AMTNR1BSLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed