SCHEMBL11083337

SCHEMBL11083337

CNCC(CN)c1cccc(OC(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
NSD2 O96028 1/20 0.43
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTT P42858 1/20 0.41
AOC3 Q16853 1/20 0.38
SLC6A4 P31645 6/20 0.38
CYP2D6 P10635 4/20 0.38
SLC6A2 P23975 4/20 0.38
SLC6A3 Q01959 4/20 0.38
KCNH2 Q12809 4/20 0.38
CYP3A4 P08684 3/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
DHFR P00374 1/20 0.38
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
PLAU P00749 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080697 0.85 AOC3 (0.54) KDM4EAOC3SLC6A4CYP2D6SLC6A2
SCHEMBL11069017 0.82 CYP3A4 (0.46) KDM4EALDH1A1AOC3SLC6A4CYP2D6
SCHEMBL11085320 0.80 KDM4E (0.42) KDM4EDHFR
SCHEMBL11084835 0.80 SLC6A3 (0.42) KDM4ESLC6A4CYP2D6SLC6A2SLC6A3
SCHEMBL25101091 0.79 HTT (0.61) KDM4ENSD2ALDH1A1SMN1; SMN2HTT
SCHEMBL11081698 0.78 BCHE (0.53) SMN1; SMN2SLC6A4CYP2D6SLC6A2SLC6A3
SCHEMBL1471425 0.76 SMN1; SMN2 (0.41) KDM4ENSD2ALDH1A1SMN1; SMN2HTT
SCHEMBL11079803 0.76 SLC6A2 (0.43) KDM4EAOC3SLC6A4CYP2D6SLC6A2
SCHEMBL18713611 0.76 ACHE (0.43) KDM4ENSD2ALDH1A1SMN1; SMN2HTT
SCHEMBL11283326 0.75 SLC6A2 (0.47) AOC3SLC6A4SLC6A2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed