SCHEMBL11080869

SCHEMBL11080869

CNCC(CN)c1ccccc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.40
ACP3 P15309 1/20 0.39
CNR2 P34972 2/20 0.38
ALDH1A1 P00352 2/20 0.36
POLB P06746 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
P2RX7 Q99572 1/20 0.35
MC4R P32245 1/20 0.35
IDO1 P14902 3/20 0.34
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
MAPK1 P28482 2/20 0.33
HSD11B1 P28845 1/20 0.33
TDO2 P48775 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087481 0.84 HTR2C (0.42) SLC6A4ACP3CNR2ALDH1A1POLB
SCHEMBL11080775 0.78 SLC6A2 (0.43) SLC6A4IDO1TDO2ADRB1ADRA2A
SCHEMBL256793 0.78 ACP3 (0.41) SLC6A4ACP3CNR2ALDH1A1POLB
Hydrochloric Acid SCHEMBL167168 0.78 CNR2 (0.46) ACP3CNR2POLB
Hydrochloric Acid SCHEMBL175643 0.77 HTR2C (0.41) SLC6A4ACP3CNR2ALDH1A1POLB
SCHEMBL11084923 0.76 TAAR1 (0.40) SLC6A4HTR2CHTR2BNOS3NOS1
SCHEMBL11080520 0.76 SLC6A2 (0.43) SLC6A4ALDH1A1ADRB1ADRA2AADRB3
SCHEMBL13703411 0.75 CNR2 (0.43) ACP3CNR2ALDH1A1POLBMAPK1
SCHEMBL11085933 0.75 NISCH (0.50) SLC6A4IDO1TDO2ADRB1CYP3A4
SCHEMBL11083546 0.75 ADRA2A (0.46) SLC6A4ALDH1A1POLBTDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed