SCHEMBL11080873

SCHEMBL11080873

CN(C)C=C(C(=O)c1ccc(Cl)cc1Cl)n1cncn1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.73
LMNA P02545 5/20 0.73
MAPT P10636 4/20 0.73
MEN1 O00255 2/20 0.73
KMT2A Q03164 2/20 0.73
CYP19A1 P11511 2/20 0.70
HTT P42858 1/20 0.67
HPGD P15428 2/20 0.53
PKM P14618 2/20 0.53
HSP90AA1 P07900 1/20 0.53
MAPK1 P28482 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
RAB9A P51151 1/20 0.48
ATM Q13315 1/20 0.48
POLB P06746 1/20 0.48
GLA P06280 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
GABRA1 P14867 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11150916 1.00 ALDH1A1 (0.73) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL11087066 0.83 CYP19A1 (0.67) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL11087065 0.83 CYP19A1 (0.67) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL10946345 0.83 CYP19A1 (0.67) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL10946350 0.83 CYP19A1 (0.67) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL8035724 0.81 MAPT (0.71) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL11298296 0.81 MAPT (0.71) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL5091820 0.81 MAPT (0.50) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL11089114 0.80 CYP19A1 (0.62) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL11089118 0.80 CYP19A1 (0.62) ALDH1A1LMNAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4435411-A Combating fungi with 1-phenyl-2-(1,2,4-triazol-1-yl)-prop-2-en-1-ones BAYER AKTIENGESELLSCHAFT (DE) 1984-03-06 US disclosed
US-4380628-A REACTING THE KETO-ENAMINE-SUBSTITUTED IMIDAZOLE OR 1,2,4-TRIAZOLE DERIVATIVE WITH A GINR ARD REAGENT; FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1983-04-19 US disclosed
EP-0032239-B1 METHOD FOR PREPARING AZOLYL-VINYL-KETONES BAYER AG (DE) 1983-01-12 EP disclosed
EP-0040367-A1 Substituted phenyl-triazolyl-vinyl ketones, process for their preparation and their application as fungicides BAYER AG (DE) 1981-11-25 EP disclosed
EP-0032239-A1 Method for preparing azolyl-vinyl-ketones BAYER AG (DE) 1981-07-22 EP disclosed