SCHEMBL11083115

SCHEMBL11083115

CNC(c1cc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)s1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.48
PTGS1 P23219 5/20 0.48
MAPK14 Q16539 7/20 0.41
KDM4E B2RXH2 1/20 0.41
MT-CO1 P00395 1/20 0.41
MT-CO2 P00403 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080131 0.78 PTGS2 (0.52) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11183966 0.78 PTGS2 (0.59) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11189076 0.77 PTGS2 (0.54) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11188282 0.75 PTGS2 (0.56) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11220738 0.74 PTGS2 (0.52) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL8985334 0.73 PTGS2 (0.50) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11191447 0.72 PTGS2 (0.50) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11087506 0.72 PTGS1 (0.51) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11182987 0.72 PTGS2 (0.52) PTGS2PTGS1MAPK14KDM4EMT-CO1
SCHEMBL11178747 0.71 PTGS2 (0.49) PTGS2PTGS1MAPK14KDM4EMT-CO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4427693-A ANTIARTHRITIC AGENTS; ANALGESICS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-01-24 US disclosed
EP-0055471-A1 Antiinflammatory 4,5-diaryl-alpha,alpha-bis(polyhalomethyl)-2-thiophenemethanamines E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-07-07 EP disclosed