SCHEMBL11083798

SCHEMBL11083798

Cc1ccccc1/C=C1\CCn2c1nc1ccc(Cl)cc1c2=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
CYP1A1 P04798 2/20 0.56
CYP1B1 Q16678 2/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 4/20 0.55
KMT2A Q03164 4/20 0.55
CCR3 P51677 5/20 0.54
ALOX5 P09917 2/20 0.51
POLB P06746 1/20 0.48
HPGD P15428 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11083801 1.00 CYP1A2 (0.56) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11084863 0.92 MEN1 (0.65) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11084861 0.92 MEN1 (0.65) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11090753 0.89 MEN1 (0.58) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11090749 0.89 MEN1 (0.58) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11089408 0.88 MEN1 (0.68) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11089405 0.88 MEN1 (0.68) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11090599 0.87 MEN1 (0.67) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11090598 0.87 MEN1 (0.67) CYP1A2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL11087084 0.87 RAB9A (0.61) CYP1A2NPC1RAB9ACYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4428952-A Substituted pyrrolo[2,1-b]quinazolines and pyrido[2,1-b]quinazolines useful for the treatment of or the prevention of gastrointestinal ulcers FARMITALIA CARLO ERBA S.P.A. (IT) 1984-01-31 US disclosed