SCHEMBL11084013

SCHEMBL11084013

NC(=O)c1ccc2nc3n(c(=O)c2c1)CC/C3=C\c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 10/20 0.59
MEN1 O00255 9/20 0.59
RAB9A P51151 3/20 0.56
NPC1 O15118 2/20 0.56
ALOX5 P09917 2/20 0.55
MAPT P10636 3/20 0.55
KDM4E B2RXH2 1/20 0.55
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 2/20 0.51
POLB P06746 1/20 0.51
THRB P10828 1/20 0.51
HPGD P15428 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MCL1 Q07820 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11084031 1.00 KMT2A (0.59) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11086734 0.94 POLB (0.57) KMT2AMEN1RAB9ANPC1MAPT
SCHEMBL11086731 0.94 POLB (0.57) KMT2AMEN1RAB9ANPC1MAPT
SCHEMBL11089854 0.93 KMT2A (0.70) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11089858 0.93 KMT2A (0.70) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11080439 0.91 KMT2A (0.70) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11080441 0.91 KMT2A (0.70) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11080382 0.89 MEN1 (0.60) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11080381 0.89 MEN1 (0.60) KMT2AMEN1RAB9ANPC1ALOX5
SCHEMBL11091304 0.86 POLB (0.66) KMT2AMEN1RAB9AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4428952-A Substituted pyrrolo[2,1-b]quinazolines and pyrido[2,1-b]quinazolines useful for the treatment of or the prevention of gastrointestinal ulcers FARMITALIA CARLO ERBA S.P.A. (IT) 1984-01-31 US disclosed