SCHEMBL11080439

SCHEMBL11080439

O=C(O)c1ccc2nc3n(c(=O)c2c1)CC/C3=C\c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.70
MEN1 O00255 8/20 0.70
MAPT P10636 2/20 0.62
RAB9A P51151 2/20 0.62
KDM4E B2RXH2 1/20 0.62
ALDH1A1 P00352 2/20 0.60
POLB P06746 2/20 0.60
HPGD P15428 2/20 0.60
THRB P10828 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
NPSR1 Q6W5P4 2/20 0.58
MCL1 Q07820 1/20 0.58
ALOX5 P09917 2/20 0.57
NPC1 O15118 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080441 1.00 KMT2A (0.70) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11088064 0.94 POLB (0.65) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11088059 0.94 POLB (0.65) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11083582 0.92 KMT2A (0.82) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11083586 0.92 KMT2A (0.82) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11080652 0.91 KMT2A (0.71) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11080648 0.91 KMT2A (0.71) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11084013 0.91 KMT2A (0.59) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11084031 0.91 KMT2A (0.59) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL11089193 0.91 KMT2A (0.65) KMT2AMEN1MAPTRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4428952-A Substituted pyrrolo[2,1-b]quinazolines and pyrido[2,1-b]quinazolines useful for the treatment of or the prevention of gastrointestinal ulcers FARMITALIA CARLO ERBA S.P.A. (IT) 1984-01-31 US claimed
US-4428952-A Substituted pyrrolo[2,1-b]quinazolines and pyrido[2,1-b]quinazolines useful for the treatment of or the prevention of gastrointestinal ulcers FARMITALIA CARLO ERBA S.P.A. (IT) 1984-01-31 US disclosed