SCHEMBL11085539

SCHEMBL11085539

CCCN1CC[C@@H](CC(O)Cc2ccnc3ccc(OC)cc23)[C@@H](CC)C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.48
KCNH2 Q12809 4/20 0.48
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 3/20 0.48
HSD17B10 Q99714 3/20 0.48
TSHR P16473 1/20 0.48
MEN1 O00255 1/20 0.48
CYP3A4 P08684 1/20 0.48
KMT2A Q03164 1/20 0.48
CHRM2 P08172 1/20 0.48
ADRA2A P08913 1/20 0.48
SLC6A4 P31645 1/20 0.48
OPRM1 P35372 1/20 0.48
SLC6A3 Q01959 1/20 0.48
ROCK2 O75116 1/20 0.46
CCR8 P51685 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976574 0.93 CCR8 (0.49) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6976570 0.93 CCR8 (0.49) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6977253 0.86 CCR8 (0.48) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL11079444 0.82 MTNR1A (0.45) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL7081967 0.82 CCR8 (0.47) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6977177 0.80 CCR8 (0.53) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6977174 0.80 CCR8 (0.53) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6977170 0.80 CCR8 (0.53) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6965276 0.78 CCR8 (0.53) CYP2D6KCNH2KDM4EALDH1A1HPGD
SCHEMBL6971729 0.77 CCR8 (0.52) CYP2D6KCNH2KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4472403-A Quinoline derivatives and pharmaceutical compositions and methods for treating cardiovascular disease with such compounds A.C.F. CHEMIEFARMA N.V. (NL) 1984-09-18 US disclosed
EP-0030044-A1 Quinoline derivatives, processes for their preparation, their use, pharmaceutical compositions containing them and a method for the preparation of these pharmaceutical compositions ACF CHEMIEFARMA NV (NL) 1981-06-10 EP disclosed