SCHEMBL11087007

SCHEMBL11087007

COC(=O)CCN(Cc1ccccc1)CC(C)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HDAC3 O15379 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
NCOR2 Q9Y618 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
MEP1B Q16820 1/20 0.41
HPGD P15428 1/20 0.40
CA12 O43570 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
LTA4H P09960 1/20 0.39
PTGES O14684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16916475 0.91 TDP1 (0.46) KDM4ETDP1ALDH1A1LMNAMEN1
SCHEMBL5175327 0.85 TDP1 (0.54) KDM4ETDP1ALDH1A1LMNAMEN1
SCHEMBL3258895 0.85 TDP1 (0.54) KDM4ETDP1ALDH1A1LMNAHDAC3
SCHEMBL21480168 0.85 KDM4E (0.46) KDM4ETDP1ALDH1A1LMNAMEN1
SCHEMBL12358653 0.83 TDP1 (0.52) KDM4ETDP1ALDH1A1LMNAMEN1
SCHEMBL10392751 0.82 ALOX5 (0.47) KDM4ETDP1ALDH1A1LMNAMEN1
SCHEMBL31301729 0.80 HDAC3 (0.52) KDM4ETDP1ALDH1A1LMNAHDAC3
SCHEMBL9332283 0.79 ALOX5 (0.49) KDM4ETDP1ALDH1A1LMNAMEN1
SCHEMBL12450937 0.78 HDAC1 (0.41) TDP1HDAC3HDAC1HDAC2NCOR2
SCHEMBL25473056 0.77 HDAC3 (0.55) KDM4ETDP1ALDH1A1LMNAHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106458996-B Fused pyrimidines as inhibitors of the p97 complex 克里弗生物科学公司 2020-11-03 CN disclosed
US-4481360-A 4H-1,2,4-Triazol-3-yl compounds THE UPJOHN COMPANY (US) 1984-11-06 US disclosed