SCHEMBL11089995

SCHEMBL11089995

CN(C)c1ccc([N+](=O)[O-])cc1CCl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
TSHR P16473 2/20 0.45
CYP19A1 P11511 10/20 0.44
HTT P42858 2/20 0.43
TP53 P04637 1/20 0.43
PDE2A O00408 1/20 0.43
PDE5A O76074 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
NFKB1 P19838 1/20 0.43
APEX1 P27695 1/20 0.43
PDE4A P27815 1/20 0.43
BLM P54132 1/20 0.43
PDE1B Q01064 1/20 0.43
PMP22 Q01453 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4D Q08499 1/20 0.43
PDE7A Q13946 1/20 0.43
PDE1C Q14123 1/20 0.43
PDE7B Q9NP56 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532457 0.85 ALDH1A1 (0.55) ALDH1A1TSHRCYP19A1HTTTP53
SCHEMBL6278023 0.83 ALDH1A1 (0.54) ALDH1A1TSHRCYP19A1HTTTP53
SCHEMBL28886071 0.83 ALDH1A1 (0.58) ALDH1A1TSHRCYP19A1HTTTP53
SCHEMBL12427118 0.81 ALDH1A1 (0.51) ALDH1A1CYP19A1HTTTP53
SCHEMBL6890955 0.78 ALDH1A1 (0.56) ALDH1A1TSHRCYP19A1HTTTP53
SCHEMBL27493611 0.78 ALDH1A1 (0.60) ALDH1A1CYP19A1HTTTP53MAPT
SCHEMBL792517 0.78 ALDH1A1 (0.49) ALDH1A1CYP19A1HTTTP53MAPT
SCHEMBL11819145 0.78 ALDH1A1 (0.64) ALDH1A1TSHRCYP19A1HTTTP53
SCHEMBL6681084 0.77 POLB (0.52) ALDH1A1TSHRHTTCYP3A4MEN1
SCHEMBL29796062 0.77 ALDH1A1 (0.60) ALDH1A1TSHRCYP19A1HTTPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4455311-A Imidazoquinazoline derivatives which inhibit the aggregation of blood platelets, inhibit gastric secretion or have activity on the circulatory system HOFFMANN-LA ROCHE INC. (US) 1984-06-19 US disclosed
EP-0073060-A1 Imidazoquinazoline derivatives, their preparation and medicaments containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-03-02 EP disclosed