SCHEMBL11090704

SCHEMBL11090704

Cc1nnc2c(c1S)CN(C(=O)c1ccccc1)CC2

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.50
MTHFD2 P13995 5/20 0.48
PTGDR2 Q9Y5Y4 4/20 0.44
CYP2C9 P11712 1/20 0.42
GRM5 P41594 2/20 0.42
KIF11 P52732 1/20 0.40
TACR3 P29371 1/20 0.40
HPGD P15428 1/20 0.40
CFTR P13569 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090495 0.84 PTGS1 (0.47) PTGS1MTHFD2PTGDR2CYP2C9CFTR
SCHEMBL11092323 0.81 CDK1 (0.50) PTGS1MTHFD2PTGDR2CYP2C9
SCHEMBL11400880 0.80 PTGS1 (0.50) PTGS1MTHFD2PTGDR2CYP2C9GRM5
SCHEMBL11397662 0.77 PTGS1 (0.58) PTGS1MTHFD2PTGDR2CYP2C9GRM5
SCHEMBL11088651 0.74 PTGS1 (0.68) PTGS1GRM5HPGD
SCHEMBL8240452 0.72 TSHR (0.49) MTHFD2PTGDR2CYP2C9GRM5HPGD
SCHEMBL12320789 0.71 KCNK3 (0.60) MTHFD2TACR3HPGD
SCHEMBL14591322 0.70 PTGDR2 (0.58) MTHFD2PTGDR2CYP2C9KIF11HPGD
SCHEMBL12680944 0.69 GRM5 (0.60) MTHFD2GRM5
SCHEMBL11085211 0.69 PTGS1 (0.68) PTGS1GRM5HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478837-A HYPOTENSIVE AGENTS SANDOZ LTD. (CH) 1984-10-23 US disclosed
US-3954754-A ANTIHYPERTENSIVES SANDOZ LTD. (CH) 1976-05-04 US disclosed