SCHEMBL11090495

SCHEMBL11090495

CCc1nnc2c(c1S)CN(C(=O)c1ccccc1)CC2

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.47
MTHFD2 P13995 4/20 0.43
PTGDR2 Q9Y5Y4 8/20 0.42
CYP2C9 P11712 2/20 0.42
BLM P54132 1/20 0.42
KCNK3 O14649 2/20 0.41
KCNK9 Q9NPC2 1/20 0.41
PTGER2 P43116 1/20 0.40
PTGDR Q13258 1/20 0.40
CFTR P13569 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11092323 0.87 CDK1 (0.50) PTGS1MTHFD2PTGDR2CYP2C9KCNK3
SCHEMBL11090704 0.84 PTGS1 (0.50) PTGS1MTHFD2PTGDR2CYP2C9CFTR
SCHEMBL11087511 0.78 LMNA (0.40) PTGDR2BLM
SCHEMBL11088759 0.76 ADORA3 (0.43) CYP2C9
Ether SCHEMBL11832353 0.75 HTR2C (0.38) CYP2C9
SCHEMBL11400880 0.75 PTGS1 (0.50) PTGS1MTHFD2PTGDR2CYP2C9KCNK3
SCHEMBL11397662 0.72 PTGS1 (0.58) PTGS1MTHFD2PTGDR2CYP2C9KCNK3
SCHEMBL12386800 0.72 PTGDR2 (0.49) MTHFD2PTGDR2CYP2C9BLMKCNK3
SCHEMBL11088651 0.72 PTGS1 (0.68) PTGS1
SCHEMBL10313025 0.70 PTGS1 (0.47) PTGS1MTHFD2PTGDR2CYP2C9BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478837-A HYPOTENSIVE AGENTS SANDOZ LTD. (CH) 1984-10-23 US disclosed
US-3954754-A ANTIHYPERTENSIVES SANDOZ LTD. (CH) 1976-05-04 US disclosed