SCHEMBL11095322

SCHEMBL11095322

Nc1cccnc1Nc1ccccc1-c1c(F)cccc1C=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
MAPK14 Q16539 2/20 0.35
ERN1 O75460 2/20 0.34
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11201136 0.89 CA12 (0.39) MAPTHTTALDH1A1SMN1; SMN2CA12
SCHEMBL11160842 0.87 KMT2A (0.37) ALDH1A1SMN1; SMN2CA12CA1CA2
SCHEMBL11122670 0.86 SMN1; SMN2 (0.43) MAPTHTTALDH1A1SMN1; SMN2CA12
SCHEMBL11154277 0.84 MEN1 (0.36) MAPTHTTSMN1; SMN2CA12CA1
SCHEMBL10370951 0.84 CA12 (0.42) MAPTHTTALDH1A1SMN1; SMN2CA12
SCHEMBL11156277 0.81 KMT2A (0.46) MAPTHTTALDH1A1SMN1; SMN2
SCHEMBL11156567 0.81 TRIM24 (0.40) MAPTHTTALDH1A1SMN1; SMN2CA12
SCHEMBL11158224 0.81 CA12 (0.38) MAPTHTTSMN1; SMN2CA12CA1
SCHEMBL11087998 0.81 KMT2A (0.40) MAPTHTTALDH1A1SMN1; SMN2CA12
SCHEMBL10373647 0.81 CA12 (0.46) MAPTHTTALDH1A1SMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0107261-A2 (2-((Nitropyridinyl)amino)phenyl)arylmethanones and salts, their use in medicine, pharmaceutical compositions containing them and their use in the preparation of (2-((aminopyridinyl)amino)phenyl)arylmethanones and pyrido(1,4)benzodiazepines A.H. ROBINS COMPANY, INCORPORATED (US) 1984-05-02 EP disclosed