SCHEMBL11101682

SCHEMBL11101682

NOCC=Cc1cccc(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.61
CYP3A4 P08684 2/20 0.50
AGXT P21549 2/20 0.50
RELA Q04206 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
GRIK1 P39086 1/20 0.47
GRIK2 Q13002 1/20 0.47
FBP1 P09467 1/20 0.45
CHAT P28329 1/20 0.45
CHRM5 P08912 1/20 0.44
GRIN1 Q05586 3/20 0.44
GRIN2B Q13224 3/20 0.44
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
NFE2L2 Q16236 3/20 0.42
AKR1C3 P42330 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11101680 1.00 IDO1 (0.61) IDO1CYP3A4AGXTRELACYP1A2
SCHEMBL7697733 0.82 RELA (0.47) IDO1RELACYP1A2CYP2C9GRIK1
SCHEMBL2771402 0.79 CYP1A2 (0.52) IDO1CYP3A4AGXTRELACYP1A2
SCHEMBL2771404 0.79 CYP1A2 (0.52) IDO1CYP3A4AGXTRELACYP1A2
SCHEMBL2097935 0.79 RELA (0.45) RELACYP1A2CYP2C9GRIK1GRIK2
SCHEMBL2097937 0.79 RELA (0.45) RELACYP1A2CYP2C9GRIK1GRIK2
SCHEMBL11128111 0.79 IDO1 (0.61) IDO1RELAFBP1MAOB
SCHEMBL11110560 0.79 IDO1 (0.61) IDO1CYP3A4AGXTRELACYP1A2
SCHEMBL11128107 0.79 IDO1 (0.61) IDO1RELAFBP1MAOB
SCHEMBL11110559 0.79 IDO1 (0.61) IDO1CYP3A4AGXTRELACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4425360-A Pharmacologically active novel O-substituted pyruvic acid oximes BOEHRINGER MANNHEIM GMBH (DE) 1984-01-10 US disclosed
EP-0048911-A2 O-substituted oximes of alpha-ketocarboxylic acid, preparation and pharmaceutical compositions Roche Diagnostics GmbH (DE) 1982-04-07 EP disclosed