SCHEMBL11112652

SCHEMBL11112652

C/C=C(\c1ccc(Br)cc1)C(c1ccc(OCCN(C)C)cc1)c1cccc(O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.48
CHRNA4 P43681 1/20 0.48
ESRRG P62508 6/20 0.43
ESRRB O95718 5/20 0.42
ESR1 P03372 7/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11133248 0.91 CHRNB2 (0.49) CHRNB2CHRNA4ESRRGESRRBESR1
SCHEMBL4309220 0.91 CHRNB2 (0.51) CHRNB2CHRNA4ESRRGESRRBESR1
SCHEMBL4309222 0.91 CHRNB2 (0.51) CHRNB2CHRNA4ESRRGESRRBESR1
SCHEMBL28421381 0.89 ESRRG (0.53) ESRRGESRRBESR1ALDH1A1LMNA
SCHEMBL2710225 0.81 CYP2D6 (0.55) ESRRGESRRBESR1KDM4EALDH1A1
SCHEMBL8732737 0.81 CYP2D6 (0.55) ESRRGESRRBESR1KDM4EALDH1A1
SCHEMBL7929087 0.81 CYP2D6 (0.55) ESRRGESRRBESR1KDM4EALDH1A1
SCHEMBL11117215 0.81 ESR1 (0.47) ESR1KDM4EALDH1A1KMT2AESR2
SCHEMBL4543424 0.80 ESR1 (0.59) ESRRGESRRBESR1KDM4EALDH1A1
SCHEMBL11570305 0.79 ESR1 (0.49) ESRRGESRRBESR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0107208-A1 1,1,2-Triphenyl-but-1-ene derivatives, process for their preparation and their use as medicines Klinge Pharma GmbH (DE) 1984-05-02 EP disclosed