SCHEMBL1111276

SCHEMBL1111276

[NH]CCc1cccc(C(F)(F)F)n1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.41
MBOAT4 Q96T53 1/20 0.38
NOTUM Q6P988 1/20 0.37
ADRB1 P08588 1/20 0.36
IDH1 O75874 4/20 0.36
IDH2 P48735 2/20 0.36
KCNH2 Q12809 2/20 0.35
MAOB P27338 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
HTR2B P41595 1/20 0.35
NR3C1 P04150 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
ADORA2A P29274 1/20 0.33
GLS O94925 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL317402 0.84 P2RX7 (0.43) P2RX7MBOAT4NOTUMADRB1IDH1
SCHEMBL7035568 0.81 P2RX7 (0.41) P2RX7MBOAT4NOTUMADRB1IDH1
SCHEMBL8190474 0.81 KCNH2 (0.46) P2RX7MBOAT4NOTUMADRB1IDH1
SCHEMBL25402832 0.81 P2RX7 (0.45) P2RX7MBOAT4NOTUMADRB1IDH1
SCHEMBL27983844 0.81 P2RX7 (0.41) P2RX7MBOAT4NOTUMADRB1IDH1
SCHEMBL23343864 0.81 P2RX7 (0.45) P2RX7MBOAT4NOTUMADRB1IDH1
SCHEMBL7037038 0.78 KCNH2 (0.43) P2RX7MBOAT4NOTUMADRB1IDH2
SCHEMBL18494297 0.78 KCNH2 (0.56) P2RX7MBOAT4ADRB1IDH1IDH2
SCHEMBL28914699 0.78 KCNH2 (0.66) P2RX7MBOAT4NOTUMKCNH2NR3C1
SCHEMBL14834464 0.78 P2RX7 (0.39) P2RX7MBOAT4NOTUMADRB1IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278968-A2 1,5-DIPHENYL-PYRROLIDIN-2-ONE COMPOUNDS AS CB-1 LIGANDS ELI LILLY AND COMPANY (US) 2011-02-02 EP disclosed