SCHEMBL11116934

SCHEMBL11116934

O=C1CCCCN1c1ccncc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
CHKA P35790 1/20 0.50
AKR1C3 P42330 5/20 0.49
HPGD P15428 4/20 0.49
DRD2 P14416 1/20 0.46
GAA P10253 1/20 0.45
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
BRD9 Q9H8M2 1/20 0.42
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696399 0.94 ALDH1A1 (0.58) ALDH1A1CHKAAKR1C3HPGDDRD2
Pyridine SCHEMBL28869905 0.86 ALDH1A1 (0.50) ALDH1A1AKR1C3HPGDGAACYP1A2
SCHEMBL31296338 0.84 ALDH1A1 (0.56) ALDH1A1AKR1C3HPGDGAAKDM4E
SCHEMBL27409503 0.80 ALDH1A1 (0.59) ALDH1A1AKR1C3HPGDCYP1A2CYP3A4
SCHEMBL76559 0.80 ALDH1A1 (0.59) ALDH1A1AKR1C3HPGDCYP1A2CYP3A4
SCHEMBL11142367 0.79 ALDH1A1 (0.74) ALDH1A1AKR1C3HPGDCYP1A2CYP3A4
SCHEMBL31500101 0.79 GAA (0.53) ALDH1A1HPGDDRD2GAACYP1A2
SCHEMBL5606442 0.79 GAA (0.53) ALDH1A1HPGDDRD2GAACYP1A2
SCHEMBL14608049 0.79 ALDH1A1 (0.46) ALDH1A1AKR1C3HPGDGAAKDM4E
SCHEMBL1626841 0.78 ALDH1A1 (0.58) ALDH1A1AKR1C3HPGDDRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0106988-A1 Pharmacologically active lactam derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-02 EP claimed
WO-2016127358-A1 INHIBITORS OF RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2016-08-18 WO disclosed
EP-1473330-B1 Process for the synthesis of oxonol compound FUJI PHOTO FILM CO LTD (JP) 2007-02-14 EP disclosed
EP-0106988-A1 Pharmacologically active lactam derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-02 EP disclosed