SCHEMBL11136754

SCHEMBL11136754

OC/C=C(/c1ccc(Cl)cc1)c1cccnc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 6/20 0.54
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALOX15 P16050 1/20 0.51
NFKB1 P19838 1/20 0.51
CYP2C19 P33261 1/20 0.51
HIF1A Q16665 1/20 0.51
ADRA2A P08913 1/20 0.51
DRD2 P14416 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
HTR2C P28335 1/20 0.51
SLC6A4 P31645 1/20 0.51
ADRA1A P35348 1/20 0.51
HRH1 P35367 1/20 0.51
OPRM1 P35372 1/20 0.51
DRD3 P35462 1/20 0.51
OPRD1 P41143 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11136755 1.00 TBXAS1 (0.54) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11136834 0.88 TBXAS1 (0.51) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11136860 0.88 TBXAS1 (0.51) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8699446 0.87 TBXAS1 (0.68) TBXAS1TBXA2R
SCHEMBL8699447 0.87 TBXAS1 (0.68) TBXAS1TBXA2R
SCHEMBL11281216 0.84 CYP3A4 (0.70) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11281219 0.84 CYP3A4 (0.70) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11143864 0.82 CYP3A4 (0.76) CYP1A2CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL11143903 0.82 CYP3A4 (0.50) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11143907 0.82 CYP3A4 (0.50) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4418065-A ANTIDEPRESSANTS ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1983-11-29 US disclosed
EP-0081478-A2 Novel halophenyl-pyridyl-allylamine derivatives, processes and intermediates as well as pharmaceutical preparations thereof Astra Läkemedel Aktiebolag (SE) 1983-06-15 EP disclosed