SCHEMBL11142402

SCHEMBL11142402

CS(=O)(=O)Nc1cc2c(cc1Oc1ccc(F)cc1F)C(=NO)CC2

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.74
PTGS1 P23219 1/20 0.46
BRD4 O60885 10/20 0.41
MAPK14 Q16539 1/20 0.41
EP300 Q09472 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11142400 1.00 PTGS2 (0.74) PTGS2PTGS1BRD4MAPK14EP300
Flosulide SCHEMBL29454969 0.85 PTGS2 (1.00) PTGS2PTGS1BRD4MAPK14
Flosulide SCHEMBL29383035 0.85 PTGS2 (1.00) PTGS2PTGS1BRD4MAPK14
Flosulide SCHEMBL195509 0.85 PTGS2 (1.00) PTGS2PTGS1BRD4MAPK14
SCHEMBL11176908 0.81 PTGS2 (0.54) PTGS2PTGS1BRD4
SCHEMBL11176910 0.81 PTGS2 (0.54) PTGS2PTGS1BRD4
SCHEMBL10935984 0.80 PTGS2 (0.71) PTGS2PTGS1BRD4MAPK14EP300
SCHEMBL10953840 0.77 PTGS2 (0.67) PTGS2PTGS1BRD4EP300
SCHEMBL10955991 0.77 PTGS2 (0.70) PTGS2PTGS1BRD4MAPK14
SCHEMBL11177616 0.76 PTGS2 (0.49) PTGS2PTGS1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4375479-A ANTIINFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 1983-03-01 US disclosed
EP-0056956-A2 Indanyl derivatives their preparation and their use SCHERING AKTIENGESELLSCHAFT (DE) 1982-08-04 EP disclosed