SCHEMBL1114372

SCHEMBL1114372

O=C1CN(C(=O)OCc2ccccc2)[C@H](c2ccc(I)cc2)O1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44
F2 P00734 2/20 0.42
ELANE P08246 2/20 0.42
CTSG P08311 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
USP2 O75604 1/20 0.41
HTR2C P28335 1/20 0.40
PDE5A O76074 1/20 0.40
PREP P48147 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28956472 0.92 PSEN1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1820197 0.77 F2 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5869413 0.77 F2 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL28956425 0.75 PSEN1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19271743 0.68 HTR2C (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL21872248 0.68 HTR2C (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6686284 0.68 SMN1; SMN2 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL30523584 0.68 HTR2C (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2011989 0.67 MEN1 (0.60) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8087093 0.67 P2RX4 (0.49) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278975-A1 NOVEL NITROSO COMPOUNDS AS NITROXYL DONORS AND METHODS OF USE THEREOF Cardioxyl Pharmaceuticals Inc. (US) 2011-02-02 EP disclosed
WO-2009137717-A1 NOVEL NITROSO COMPOUNDS AS NITROXYL DONORS AND METHODS OF USE THEREOF CARDIOXYL PHARMACEUTICALS INC. (US) 2009-11-12 WO disclosed