SCHEMBL1114657

SCHEMBL1114657

CCCCCCCCCCCCCCCC(=O)N[C@H]1CCCNC(=O)C1[C@@H]1CCC(NC(=O)CCCCCCCCCC)CC(=O)N1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.52
GNAI3 P08754 1/20 0.44
GNAO1 P09471 1/20 0.44
GNAI1 P63096 1/20 0.44
NAAA Q02083 3/20 0.43
NOD1 Q9Y239 1/20 0.43
CNR1 P21554 5/20 0.40
CNR2 P34972 5/20 0.40
TRPV1 Q8NER1 4/20 0.39
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CXCR4 P61073 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114788 1.00 CCR2 (0.52) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL5699632 1.00 CCR2 (0.52) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL5699622 1.00 CCR2 (0.52) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114631 0.95 CCR2 (0.47) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114932 0.80 CCR2 (0.60) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114962 0.80 CCR2 (0.60) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114852 0.80 CCR2 (0.60) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114672 0.80 CCR2 (0.60) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114444 0.80 CCR2 (0.60) CCR2GNAI3GNAO1GNAI1NAAA
SCHEMBL1114510 0.80 CCR2 (0.60) CCR2GNAI3GNAO1GNAI1NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279741-A2 Caprolactams and their use as anti-inflammatory agents Cambridge Enterprise Ltd. (GB) 2011-02-02 EP claimed
EP-1691814-A2 ANTI-INFLAMMATORY AGENTS CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LIMITED (GB) 2006-08-23 EP claimed
WO-2005053702-A2 ANTI-INFLAMMATORY AGENTS CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LIMITED (GB) 2005-06-16 WO claimed
EP-1691814-A2 ANTI-INFLAMMATORY AGENTS CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LIMITED (GB) 2006-08-23 EP disclosed
WO-2005053702-A2 ANTI-INFLAMMATORY AGENTS CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LIMITED (GB) 2005-06-16 WO disclosed